AX20017 does not affect the human kinases
3R)-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-2
Inupadenant has potent anti-tumor activity
Chemical Name: 4-[2-(5-amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-(1
GNE-272 is a potent and selective CBP/EP300 inhibitor with IC50 values of 0
(−)-Apomorphine (hydrochloride) Catalog No.:M22410-C AX20017 does not affect the() Apomorphine is a non selective dopamine receptor agonist that exhibits pKi values of 6. 43, 7. 08, 7. 59, 8. 36, and 7. 83 for human recombinant D1, D2L, D3, D4, and D5 receptors, respectively., It produces biphasic effects on locomotor activity and displays anti parkinsonian and neuroprotective actions.[1,], . Millan, M. J., Maiofiss, L., Cussac, D., et al. Differential actions of antiparkinson agents at multiple classes of monoaminergic receptor.